SCHEMBL9954331

SCHEMBL9954331

Fc1cccc(-c2coc(Cl)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50
ALDH1A1 P00352 1/20 0.44
IDO1 P14902 2/20 0.44
NOTUM Q6P988 1/20 0.44
KMO O15229 2/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
MAP4K4 O95819 2/20 0.40
GRM5 P41594 1/20 0.39
NT5E P21589 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
TP53 P04637 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
ESR2 Q92731 1/20 0.38
HPGDS O60760 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955528 0.82 CYP19A1 (0.46) KDM4EALDH1A1IDO1NOTUMKMO
SCHEMBL9954530 0.79 ENPP3 (0.59) KDM4EKMT2AIDO1KMOBCHE
SCHEMBL28702905 0.79 KDM4E (0.46) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL10263247 0.79 ENPP3 (0.59) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL3637967 0.78 RAB9A (0.44) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL3635042 0.77 MEN1 (0.48) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL26131327 0.77 BRD4 (0.37) MAP4K4GRM5
SCHEMBL14637364 0.77 RAB9A (0.40) KDM4EMEN1KMT2AALDH1A1NOTUM
SCHEMBL9955922 0.76 KDM4E (0.68) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL3632196 0.76 CYP19A1 (0.48) KDM4EMAPTALDH1A1NOTUMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed