SCHEMBL9956730

SCHEMBL9956730

Cc1ccc2c(Br)cc(Br)c(Oc3ccccc3CC=O)c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
LMNA P02545 3/20 0.37
HTT P42858 2/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 4/20 0.34
POLB P06746 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
USP2 O75604 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
PKM P14618 1/20 0.33
NQO2 P16083 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956727 0.77 PARP1 (0.37) KDM4ELMNAHTTKMT2AMEN1
SCHEMBL7690476 0.70 NQO2 (0.50) KDM4ELMNAHTTKMT2AMEN1
SCHEMBL9951347 0.69 KDM4E (0.41) KDM4ELMNAHTTKMT2AMEN1
Broxaldine SCHEMBL2109050 0.68 ALOX5 (0.41) KDM4ELMNAHTTKMT2AMEN1
Broxaldine SCHEMBL29888411 0.68 ALOX5 (0.41) KDM4ELMNAHTTKMT2AMEN1
SCHEMBL2167807 0.68 CXCL8 (0.42) KDM4ELMNAHTTKMT2AMAPT
SCHEMBL9951316 0.68 KDM4E (0.49) KDM4ELMNAHTTKMT2AMEN1
SCHEMBL28554817 0.67 KDM4E (0.40) KDM4ELMNAHTTKMT2AMEN1
SCHEMBL18106122 0.67 KDM4E (0.42) KDM4EHTTKMT2AMEN1MAPT
SCHEMBL1461233 0.64 KMT2A (0.56) KDM4ELMNAHTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083866-A1 QUINOLINE DERIVATIVES AS ANTI-CANCER AGENTS THE HONG KONG POLYTECHNIC UNIVERSITY (CN) 2012-06-28 WO disclosed