SCHEMBL9957231

SCHEMBL9957231

Nc1nc2c(c(=O)[nH]1)C=CCN2

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 8/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
PMP22 Q01453 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PNP P00491 2/20 0.36
QTRT1 Q9BXR0 1/20 0.35
NOS3 P29474 2/20 0.35
NOS2 P35228 2/20 0.35
DYRK1A Q13627 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956185 0.69 TYMS (0.41) PNP
SCHEMBL676634 0.69 KDM4E (0.43) NOS1KDM4ELMNAHSD17B10PNP
Hydrochloric Acid SCHEMBL9545316 0.66 XDH (0.33) NOS1KDM4EHSD17B10PNPQTRT1
SCHEMBL9793234 0.64 PLAUR (0.37) KDM4EALDH1A1PMP22HSD17B10
SCHEMBL3454164 0.63 NOS1 (0.53) NOS1KDM4EALDH1A1LMNAGLA
SCHEMBL9544092 0.63 TYMS (0.34) NOS1QTRT1
SCHEMBL9544423 0.63 HSD17B10 (0.33) KDM4EHSD17B10PNPQTRT1
SCHEMBL9545341 0.61 PNP (0.35) NOS1PNPQTRT1
SCHEMBL17556623 0.60 NOS1 (0.49) NOS1KDM4EALDH1A1LMNAGLA
SCHEMBL3454196 0.59 NOS1 (0.41) NOS1KDM4EALDH1A1LMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed