SCHEMBL9958481

SCHEMBL9958481

COc1ccc(C)cc1S(=O)(=O)Nc1ccc2c(c1)CCN(OC(=O)OC(C)(C)C)C2

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TRIM24 O15164 10/20 0.50
LMNA P02545 3/20 0.50
HPGD P15428 3/20 0.50
THRB P10828 1/20 0.46
ALDH1A1 P00352 1/20 0.46
BRPF1 P55201 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3156959 0.85 SMN1; SMN2 (0.54) SMN1; SMN2MEN1KMT2ATRIM24LMNA
SCHEMBL9959634 0.80 MAPT (0.50) SMN1; SMN2KMT2ATRIM24LMNAALDH1A1
SCHEMBL9960391 0.79 ALDH1A1 (0.45) TRIM24ALDH1A1
SCHEMBL9959434 0.78 NLRP3 (0.51) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL9958499 0.78 NAMPT (0.47) KMT2ATRIM24
SCHEMBL9958328 0.75 HTR6 (0.53) NPSR1
SCHEMBL9957615 0.74 HTR6 (0.53)
SCHEMBL10240546 0.73 ESR2 (0.54) SMN1; SMN2LMNATHRBALDH1A1NPSR1
SCHEMBL13757743 0.72 SMN1; SMN2 (0.62) SMN1; SMN2MEN1KMT2ALMNAHPGD
SCHEMBL7284689 0.72 ESR2 (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081600-B1 Combination of the NMDA- receptor ligand memantine and a compound with 5-HT6 receptor affinity ESTEVE LABOR DR (ES) 2012-12-05 EP claimed
EP-2007729-B1 SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS ESTEVE LABOR DR (ES) 2012-06-27 EP claimed