SCHEMBL9959634

SCHEMBL9959634

Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN(OC(=O)OC(C)(C)C)C3)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
TRIM24 O15164 3/20 0.42
RORC P51449 1/20 0.40
LMNA P02545 3/20 0.38
KCNA1 Q09470 2/20 0.38
KCNAB1 Q14722 2/20 0.38
RECQL P46063 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NR3C1 P04150 1/20 0.38
FABP4 P15090 4/20 0.37
FABP5 Q01469 1/20 0.37
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9960391 0.88 ALDH1A1 (0.45) TRIM24RORCALDH1A1BRD4
SCHEMBL3142771 0.85 ESR2 (0.53) MAPTTRIM24LMNAKCNA1KCNAB1
SCHEMBL9959434 0.82 NLRP3 (0.51) MAPTLMNAKCNA1KCNAB1ALDH1A1
SCHEMBL9958481 0.80 SMN1; SMN2 (0.52) TRIM24LMNANPSR1ALDH1A1SMN1; SMN2
SCHEMBL5242130 0.80 MAPT (0.51) MAPTTRIM24RORCLMNAKCNA1
SCHEMBL9958499 0.79 NAMPT (0.47) TRIM24KCNA1KCNAB1CYP1A2CYP3A4
SCHEMBL13757713 0.79 DRD2 (0.50) MAPTLMNAKCNA1KCNAB1NPSR1
Hydrochloric Acid SCHEMBL3147505 0.78 DRD2 (0.49) MAPTLMNAKCNA1KCNAB1NPSR1
SCHEMBL10240588 0.77 DRD2 (0.51) MAPTTRIM24LMNARECQLNPSR1
SCHEMBL9958328 0.76 HTR6 (0.53) NPSR1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081600-B1 Combination of the NMDA- receptor ligand memantine and a compound with 5-HT6 receptor affinity ESTEVE LABOR DR (ES) 2012-12-05 EP claimed
EP-2007729-B1 SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS ESTEVE LABOR DR (ES) 2012-06-27 EP claimed