SCHEMBL9968618

SCHEMBL9968618

CCC(=O)c1cc(S(=O)(=O)NCc2ccc(O)c(O)c2)ccc1C

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
HCRTR1 O43613 1/20 0.45
RAB9A P51151 3/20 0.45
POLB P06746 3/20 0.45
NPC1 O15118 2/20 0.45
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 2/20 0.42
MEN1 O00255 1/20 0.42
CYP19A1 P11511 2/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9968477 0.84 ALDH1A1 (0.43) KMT2ARAB9APOLBKDM4EALDH1A1
SCHEMBL9968569 0.82 MAPK1 (0.44) KMT2ARAB9APOLBKDM4EALDH1A1
SCHEMBL9941581 0.81 KMT2A (0.63) KMT2APOLBALDH1A1HPGDMEN1
SCHEMBL9968476 0.74 ALDH1A1 (0.47) POLBKDM4EALDH1A1HPGDMAPK1
SCHEMBL9968581 0.72 KDM4E (0.43) KMT2ARAB9APOLBKDM4EALDH1A1
SCHEMBL11517004 0.70 LMNA (0.46) KMT2ARAB9APOLBNPC1ALDH1A1
SCHEMBL6078727 0.70 CYP19A1 (0.50) KMT2APOLBMEN1CYP19A1LMNA
SCHEMBL15682651 0.69 KEAP1 (0.64) POLBKDM4EALDH1A1HPGDMAPK1
SCHEMBL9941859 0.69 MAPT (0.65) KMT2APOLBALDH1A1HPGDMEN1
SCHEMBL9941510 0.69 ALDH1A1 (0.66) KMT2APOLBALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082862-A2 ANDROGEN RECEPTOR INHIBITORS AND METHODS OF USE THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER (US) 2012-06-21 WO disclosed