SCHEMBL9969978

SCHEMBL9969978

C/C(N)=N/c1cc(C)ccc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
TDP1 Q9NUW8 4/20 0.43
GAA P10253 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
HTR3E A5X5Y0 2/20 0.40
HTR3B O95264 2/20 0.40
HTR3A P46098 2/20 0.40
HTR3D Q70Z44 2/20 0.40
HTR3C Q8WXA8 2/20 0.40
NOS1 P29475 2/20 0.40
CYP2D6 P10635 2/20 0.40
PLAU P00749 2/20 0.40
DHODH Q02127 1/20 0.40
SLC22A2 O15244 1/20 0.40
SLC22A1 O15245 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12516764 0.87 HTR3E (0.50) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL19358313 0.84 NPC1 (0.42) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL19358314 0.84 NPC1 (0.42) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL13654945 0.84 NPC1 (0.42) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL21131268 0.83 NPC1 (0.50) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL21900388 0.83 NPC1 (0.50) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL17225195 0.81 NPC1 (0.40) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL12516766 0.80 MEN1 (0.43) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL12516767 0.80 KDM4E (0.43) ALDH1A1TDP1GAAKDM4EHTT
SCHEMBL12516763 0.80 ALDH1A1 (0.44) ALDH1A1TDP1GAAKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835427-B2 Fungicidal heterocyclic compounds E I DU PONT DE NEMOURS AND COMPANY (US) 2014-09-16 US disclosed
US-8722678-B2 Fungicidal oximes and hydrazones E I DU PONT DE NEMOURS AND COMPANY (US) 2014-05-13 US disclosed
US-8722678-B2 Fungicidal oximes and hydrazones E I DU PONT DE NEMOURS AND COMPANY (US) 2014-05-13 US disclosed
US-20130261154-A1 FUNGICIDAL AZOCYCLIC AMIDES E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-03 US disclosed
US-20130261154-A1 FUNGICIDAL AZOCYCLIC AMIDES E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-03 US disclosed
US-20130030002-A1 FUNGICIDAL OXIMES AND HYDRAZONES E I DUPONT DE NEMOURS AND COMPANY (US) 2013-01-31 US disclosed
US-20130030002-A1 FUNGICIDAL OXIMES AND HYDRAZONES E I DUPONT DE NEMOURS AND COMPANY (US) 2013-01-31 US disclosed
US-20120309752-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS E I DU PONT DE NEMOURS AND COMPANY (US) 2012-12-06 US disclosed
WO-2012082580-A2 FUNGICIDAL AZOCYCLIC AMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-06-21 WO disclosed
WO-2011146182-A1 FUNGICIDAL OXIMES AND HYDRAZONES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130261154-A1 FUNGICIDAL AZOCYCLIC AMIDES CYP51A1, Q6ZSR9, NOX1 ALDH1A1 1346/4885TDP1 1802/4885GAA 139/4885
US-20120309752-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS CYP1B1, NOX3, CYP1A1 ALDH1A1 749/4885TDP1 1005/4885GAA 168/4885
US-20130030002-A1 FUNGICIDAL OXIMES AND HYDRAZONES NOX1, QSOX1, XDH ALDH1A1 418/4885TDP1 884/4885GAA 329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.