SCHEMBL9980448

SCHEMBL9980448

NS(=O)(=O)c1ccc(N2CCOCC2)c(CNc2ncnc3[nH]nc(-c4cccc(Cl)c4)c23)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.42
STK4 Q13043 3/20 0.42
STK3 Q13188 3/20 0.42
EGFR P00533 3/20 0.41
BRAF P15056 4/20 0.40
CDK2 P24941 1/20 0.38
TNNI3K Q59H18 3/20 0.38
TTK P33981 1/20 0.37
PTGS2 P35354 1/20 0.37
CDK1 P06493 2/20 0.37
SRC P12931 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CNR2 P34972 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
ABL1 P00519 1/20 0.36
PRKCA P17252 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980404 0.84 STK4 (0.39) LRRK2STK4STK3EGFRBRAF
SCHEMBL12065785 0.79 BRAF (0.67) LRRK2STK4STK3BRAFTNNI3K
SCHEMBL30295802 0.75 LRRK2 (0.67) LRRK2STK4STK3CNR2
SCHEMBL9980486 0.74 FFAR2 (0.33) LRRK2ALDH1A1CA1CA2
SCHEMBL9980436 0.73 TNNI3K (0.37) EGFRBRAFTNNI3KCA12CA1
SCHEMBL9980493 0.72 TNNI3K (0.36) LRRK2EGFRBRAFTNNI3KALDH1A1
SCHEMBL1809126 0.71 SRC (0.43) EGFRBRAFTNNI3KSRC
SCHEMBL2225236 0.71 TNNI3K (0.51) EGFRCDK2TNNI3KCDK1CA12
SCHEMBL9980391 0.70 EGFR (0.41) EGFRBRAFTNNI3KSRCALDH1A1
SCHEMBL9980424 0.70 TNNI3K (0.35) LRRK2EGFRBRAFTNNI3KCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed