SCHEMBL9980424

SCHEMBL9980424

COC1CCN(c2ccc(S(N)(=O)=O)cc2CNc2ncnc3[nH]nc(Br)c23)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 3/20 0.35
FFAR2 O15552 2/20 0.35
BRAF P15056 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA7 P43166 2/20 0.35
CA13 Q8N1Q1 2/20 0.35
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
NAMPT P43490 1/20 0.33
EGFR P00533 2/20 0.32
ERBB2 P04626 1/20 0.32
CHRM4 P08173 2/20 0.32
MAP4K4 O95819 1/20 0.32
LMNA P02545 1/20 0.32
LRRK2 Q5S007 2/20 0.31
PDE5A O76074 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
PIK3CA P42336 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980493 0.91 TNNI3K (0.36) TNNI3KFFAR2BRAFCA1CA2
SCHEMBL9980436 0.87 TNNI3K (0.37) TNNI3KBRAFCA1CA2CA7
SCHEMBL9980416 0.83 TNNI3K (0.43) TNNI3KFFAR2BRAFCA1CA2
SCHEMBL12067159 0.78 TNNI3K (0.57) TNNI3KBRAF
SCHEMBL9980486 0.76 FFAR2 (0.33) FFAR2CA1CA2CA7CA13
SCHEMBL9980375 0.73 TNNI3K (0.40) TNNI3KBRAFCA1CA2CA7
SCHEMBL9980404 0.71 STK4 (0.39) TNNI3KBRAFEGFRLMNALRRK2
SCHEMBL9980448 0.70 LRRK2 (0.42) TNNI3KBRAFCA1CA2EGFR
SCHEMBL12066468 0.69 TNNI3K (0.55) TNNI3KBRAF
SCHEMBL1809126 0.69 SRC (0.43) TNNI3KBRAFEGFRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed