SCHEMBL9983071

SCHEMBL9983071

c1ccc(COc2cccc(-c3ncc4cn[nH]c4n3)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.51
KDM4E B2RXH2 1/20 0.49
HSP90AA1 P07900 1/20 0.49
MAPT P10636 1/20 0.49
MAPK1 P28482 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CB P42338 1/20 0.47
PIK3CG P48736 1/20 0.47
PRKDC P78527 1/20 0.47
DYRK1B Q9Y463 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.45
CYP4F2 P78329 1/20 0.45
CYP4A11 Q02928 1/20 0.45
BCHE P06276 1/20 0.45
ROCK2 O75116 1/20 0.44
GRK2 P25098 1/20 0.44
NR4A2 P43354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3762000 0.78 HPGDS (0.47) HSP90AA1MAPTDYRK1BFGFR1
SCHEMBL8390694 0.77 CYP4F2 (0.56) KDM4EHSP90AA1MAPTMAPK1NPSR1
SCHEMBL8390697 0.76 MAOB (0.62) MRGPRX4CYP4F2CYP4A11BCHENR4A2
SCHEMBL379281 0.74 MAOB (0.67) MRGPRX4CYP4F2CYP4A11BCHENR4A2
SCHEMBL4051954 0.73 AKT1 (0.54) CDC7KDM4EHSP90AA1MAPTMAPK1
SCHEMBL2137838 0.73 MRGPRX4 (0.69) MRGPRX4CYP4F2CYP4A11BCHENR4A2
SCHEMBL3757242 0.73 METAP2 (0.47) DYRK1BROCK2FGFR1FGFR2FGFR3
SCHEMBL2570284 0.72 CDC7 (0.61) CDC7KDM4EHSP90AA1MAPTMAPK1
SCHEMBL29463390 0.72 ALOX5 (0.58) CDC7KDM4EHSP90AA1MAPTMAPK1
SCHEMBL4977897 0.72 ALOX5 (0.58) CDC7KDM4EHSP90AA1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8076338-B2 Such as 6-(4-phenylpiperazin-1-yl)-9H-purine; cell proliferation/differentiation EXELIXIS, INC. (US) 2011-12-13 US disclosed