Proline

Proline

SCHEMBL998686

NC(=O)O.O=C(O)[C@@H]1CCCN1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC5A2

The experimentally established mechanism targets of Proline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 3/20 0.56
NOS3 P29474 2/20 0.56
NOS1 P29475 2/20 0.56
BLM P54132 2/20 0.47
GLI1 P08151 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
DPP4 P27487 4/20 0.44
DPP8 Q6V1X1 2/20 0.44
DPP9 Q86TI2 2/20 0.44
FAP Q12884 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
SLC6A1 P30531 2/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 2/20 0.39
SLC6A11 P48066 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A13 Q9NSD5 1/20 0.39
CYP2D6 P10635 2/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Proline SCHEMBL998685 1.00 NOS2 (0.56) NOS2NOS3NOS1BLMGLI1
Proline SCHEMBL3987842 0.95 NOS2 (0.56) NOS2NOS3NOS1BLMGLI1
Proline SCHEMBL3987839 0.95 NOS2 (0.56) NOS2NOS3NOS1BLMGLI1
Proline SCHEMBL27997258 0.93 NOS2 (0.54) NOS2NOS3NOS1BLMGLI1
Pipecolic Acid SCHEMBL2263946 0.93 NOS2 (0.48) NOS2NOS3NOS1BLMGLI1
Proline SCHEMBL27694737 0.93 NOS2 (0.52) NOS2NOS3NOS1BLMGLI1
Proline SCHEMBL462226 0.93 BLM (0.52) NOS2NOS3NOS1BLMMEN1
Proline SCHEMBL10141185 0.93
Proline SCHEMBL462225 0.93 BLM (0.52) NOS2NOS3NOS1BLMMEN1
D-Proline SCHEMBL21462052 0.93 BLM (0.52) NOS2NOS3NOS1BLMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120575190-A Method for synthesizing proline carbamate by catalyzing guanidine-based porous organic polymer 广西师范大学 2025-09-02 CN disclosed
CN-120575190-A Method for synthesizing proline carbamate by catalyzing guanidine-based porous organic polymer 广西师范大学 2025-09-02 CN disclosed
US-20120270847-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIATES AND USES THEREOF SHIRE LLC (US) 2012-10-25 US disclosed
EP-2453900-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIOIDS AND USES THEREOF Shire LLC (US) 2012-05-23 EP disclosed
US-20110209227-A1 METHODS FOR THE DIAGNOSIS AND TREATMENT OF BONE DISORDERS TCP INNOVATIONS LIMITED (GB) 2011-08-25 US disclosed
US-7901873-B2 Chemometric analysis which utilizes free proline as a diagnostic and prognostic indicator of conditions associated with low bone mineral density; osteoporosis TCP INNOVATIONS LIMITED (GB) 2011-03-08 US disclosed
WO-2011007247-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIOIDS AND USES THEREOF SHIRE LLC (US) 2011-01-20 WO disclosed
US-20110015182-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIOIDS AND USES THEREOF SHIRE LLC 2011-01-20 US disclosed
US-20040241743-A1 Methods for the diagnosis and treatment of bone disorders TCP INNOVATIONS LIMITED (GB) 2004-12-02 US disclosed
EP-1384074-A2 METHODS FOR THE DIAGNOSIS AND TREATMENT OF BONE DISORDERS Metabometrix Limited (GB) 2004-01-28 EP disclosed
WO-2002086502-A2 METHODS FOR THE DIAGNOSIS AND TREATMENT OF BONE DISORDERS METABOMETRIX LIMITED (GB) 2002-10-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110015182-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIOIDS AND USES THEREOF OPRL1, OPRM1, DNPEP NOS2 213/4885NOS3 178/4885NOS1 192/4885
US-20110209227-A1 METHODS FOR THE DIAGNOSIS AND TREATMENT OF BONE DISORDERS SOST, PTH1R, COL2A1 NOS2 1342/4885NOS3 533/4885NOS1 941/4885
US-20120270847-A1 NOVEL CARBAMATE AMINO ACID AND PEPTIDE PRODRUGS OF OPIATES AND USES THEREOF OPRL1, OPRM1, DNPEP NOS2 332/4885NOS3 249/4885NOS1 266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.