SCHEMBL9987688

SCHEMBL9987688

CNC(=O)c1c(C)c2ccccc2n1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
EGFR P00533 2/20 0.41
SRC P12931 1/20 0.41
PLK1 P53350 3/20 0.41
KDM4E B2RXH2 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
F10 P00742 1/20 0.38
NR4A2 P43354 1/20 0.38
PTPN7 P35236 1/20 0.38
MAPT P10636 1/20 0.37
BRD4 O60885 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568557 0.80 TSHR (0.60) TSHREGFRSRCKDM4EL3MBTL1
SCHEMBL25433493 0.71 TSHR (0.51) TSHRKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4236344 0.71 SMN1; SMN2 (0.47) KDM4EL3MBTL1SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL4208219 0.70 KDM4E (0.62) TSHREGFRSRCKDM4EL3MBTL1
SCHEMBL1421429 0.69 CCR2 (0.51) EGFRKDM4ESMN1; SMN2ALDH1A1NR4A2
SCHEMBL1408375 0.68 SMN1; SMN2 (0.56) KDM4EL3MBTL1SMN1; SMN2ALDH1A1HPGD
SCHEMBL7607181 0.68 KMT2A (0.43) KDM4ESMN1; SMN2ALDH1A1HPGDHDAC1
SCHEMBL30234519 0.68 MCL1 (0.45) TSHRPLK1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL27527098 0.68 L3MBTL1 (0.44) TSHRKDM4EL3MBTL1ALDH1A1HSD17B10
SCHEMBL9987683 0.68 MCL1 (0.45) TSHRPLK1KDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163195-A1 FUSED PYRROLE DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-12-29 WO disclosed