SCHEMBL10033135

SCHEMBL10033135

COC(=O)CC1CCCC(N(CC2CCCCC2)CC2CCCCC2)C1c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.38
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
TAS1R2 Q8TE23 2/20 0.36
CTSD P07339 3/20 0.34
HSD11B1 P28845 1/20 0.33
FFAR1 O14842 1/20 0.33
EPHX1 P07099 1/20 0.32
PKM P14618 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CHRM3 P20309 1/20 0.32
EPHX2 P34913 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033134 0.90 USP30 (0.36) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL1709454 0.89 SLC6A2 (0.40) KCNN4SLC6A2SLC6A4TAS1R3TAS1R1
SCHEMBL10033001 0.83 NPC1 (0.38) ALDH1A1
SCHEMBL10033003 0.81 EPHX2 (0.45) EPHX2ALDH1A1
SCHEMBL1709399 0.80 PTGDR (0.41) CTSDHDAC3HDAC1HDAC2HDAC8
SCHEMBL1709398 0.78 KDM1A (0.36) CTSDEPHX1HDAC1HDAC8HDAC6
SCHEMBL1709359 0.78 USP30 (0.38) SLC6A2SLC6A4PKMHDAC3HDAC1
SCHEMBL1709374 0.75 KMT2A (0.39) ALDH1A1
SCHEMBL1709358 0.75 DPEP1 (0.36) SLC6A2SLC6A4TAS1R3TAS1R1TAS1R2
SCHEMBL10032829 0.75 FFAR1 (0.41) KCNN4TAS1R3TAS1R1TAS1R2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed