SCHEMBL10054046

SCHEMBL10054046

Cc1cc2cccc(O)c2cc1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 5/20 0.59
HSD17B2 P37059 5/20 0.59
GRIN2D O15399 1/20 0.53
GRIN2A Q12879 1/20 0.53
GRIN2B Q13224 1/20 0.53
GRIN2C Q14957 1/20 0.53
PLAU P00749 1/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
CYP1A2 P05177 3/20 0.48
ESR1 P03372 2/20 0.46
ESR2 Q92731 2/20 0.46
TLR8 Q9NR97 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
G6PD P11413 1/20 0.44
CYP2C9 P11712 1/20 0.44
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2608798 0.91 HSD17B1 (0.59) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL5083275 0.89 HSD17B1 (0.56) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL19425721 0.83 HSD17B1 (0.55) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL15631716 0.82 HSD17B1 (0.50) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL14100569 0.82 HSD17B1 (0.46) HSD17B1HSD17B2PLAUCTDSP1CYP1A2
SCHEMBL7793914 0.81 GRIN2D (0.61) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL29857010 0.81 CYP1A2 (0.62) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL2115683 0.81 CYP1A2 (0.62) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B
SCHEMBL23912230 0.79 ALDH1A1 (0.58) CYP1A2ALDH1A1MAPTHPGDHIF1A
SCHEMBL7046826 0.79 HSD17B1 (0.47) HSD17B1HSD17B2GRIN2DGRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017210072-A1 ELECTROACTIVE COMPOUNDS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2017-12-07 WO disclosed
US-8946188-B2 Anti-microbial agents and uses thereof SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2015-02-03 US disclosed
EP-2590950-B1 N-CYCLYL-3-(CYCLYLCARBONYLAMINOMETHYL)BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2014-10-15 EP disclosed
US-20140024611-A1 ANTI-MICROBIAL AGENTS AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-01-23 US disclosed
US-8461128-B2 Anti-microbial agents and uses thereof SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2013-06-11 US disclosed
US-20120165322-A1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 US disclosed
WO-2012006203-A1 N-CYCLYL-3 - (CYCLYLCARBONYLAMINOMETHYL) BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed
US-20090170805-A1 ANTI-MICROBIAL AGENTS AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140024611-A1 ANTI-MICROBIAL AGENTS AND USES THEREOF ACAT1, ACAT2, APEH HSD17B1 3947/4885HSD17B2 4223/4885GRIN2D 4171/4885
US-20120165322-A1 RHO KINASE INHIBITORS ROCK1, ROCK2, RHOA HSD17B1 1547/4885HSD17B2 1666/4885GRIN2D 4562/4885
US-20090170805-A1 ANTI-MICROBIAL AGENTS AND USES THEREOF ACAT1, ACAT2, APEH HSD17B1 3947/4885HSD17B2 4223/4885GRIN2D 4171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.