SCHEMBL10071960

SCHEMBL10071960

Clc1ccccc1CCNCC1CC12CCN(c1ccccc1)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.49
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
KCNH2 Q12809 1/20 0.36
NAMPT P43490 1/20 0.36
CXCR4 P61073 4/20 0.35
CCR3 P51677 1/20 0.35
RIPK1 Q13546 1/20 0.35
METAP2 P50579 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709237 0.80 SCN9A (0.58) SCN9ANAMPT
SCHEMBL1709243 0.77 SCN9A (0.52) SCN9AKDM4EMEN1KMT2AMAPT
SCHEMBL10071959 0.76 CCR3 (0.51) SCN9AALDH1A1MEN1KMT2AGAA
SCHEMBL1709240 0.71 SCN9A (0.60) SCN9AKDM4EALDH1A1MEN1KMT2A
SCHEMBL1709217 0.71 SCN9A (0.48) SCN9AALDH1A1KMT2AKCNH2P2RX7
SCHEMBL1709251 0.71 SCN9A (0.54) SCN9AKDM4EALDH1A1MEN1KMT2A
SCHEMBL10072038 0.68 SCN9A (0.53) SCN9AALDH1A1MEN1KMT2ACYP3A4
SCHEMBL1966295 0.68 MEN1 (0.70) MEN1KMT2ATAAR1CXCR4TP53
SCHEMBL1709241 0.67 SCN9A (0.54) SCN9AKDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL10834316 0.67 TAAR1 (0.69) MEN1KMT2ATAAR1KCNH2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed