SCHEMBL10071959

SCHEMBL10071959

COc1ccc(CCNCC2CC23CCN(c2ccccc2)CC3)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 3/20 0.51
SCN9A Q15858 1/20 0.49
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 1/20 0.44
CHRM5 P08912 2/20 0.43
CHRM3 P20309 2/20 0.43
ATM Q13315 1/20 0.43
BCHE P06276 2/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP3A4 P08684 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CHRM1 P11229 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709237 0.82 SCN9A (0.58) SCN9ASMN1; SMN2
SCHEMBL10071960 0.76 SCN9A (0.49) CCR3SCN9AMEN1KMT2AGAA
SCHEMBL1709243 0.72 SCN9A (0.52) SCN9AMEN1KMT2AUSP2CYP3A4
SCHEMBL7899024 0.70 ADRA1D (0.55) ADRA1DADRA1AADRA1BGAAALDH1A1
SCHEMBL4614753 0.69 MEN1 (0.71) MEN1KMT2AGAAATMBCHE
SCHEMBL1709217 0.69 SCN9A (0.48) SCN9AKMT2AALDH1A1
SCHEMBL10072038 0.69 SCN9A (0.53) SCN9AMEN1KMT2AUSP2ALDH1A1
SCHEMBL1709241 0.68 SCN9A (0.54) SCN9AUSP2ALDH1A1CYP3A4
SCHEMBL18840909 0.67 CCR3 (1.00) CCR3
SCHEMBL10072040 0.67 NAMPT (0.52) MEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed