SCHEMBL1709241

SCHEMBL1709241

CCCC1CC12CCN(c1ccccc1)CC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.54
SIGMAR1 Q99720 2/20 0.46
DRD2 P14416 1/20 0.46
CHRNA7 P36544 3/20 0.45
DPP4 P27487 2/20 0.43
USP2 O75604 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HTR7 P34969 3/20 0.40
HRH3 Q9Y5N1 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GFER P55789 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
CHRNB2 P17787 1/20 0.39
NFKB1 P19838 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286796 0.76 USP2 (0.49) SCN9ASIGMAR1CHRNA7USP2CYP2D6
SCHEMBL1709252 0.75 SCN9A (0.56) SCN9ASIGMAR1DRD2CHRNA7DPP4
SCHEMBL1709240 0.74 SCN9A (0.60) SCN9ASIGMAR1USP2CYP2D6ALDH1A1
SCHEMBL10072038 0.74 SCN9A (0.53) SCN9ACHRNA7USP2CYP2D6CYP2C9
SCHEMBL1709243 0.73 SCN9A (0.52) SCN9AUSP2CYP2D6KDM4ECYP3A4
SCHEMBL1709249 0.73 DRD4 (0.60) SCN9ASIGMAR1DRD2HTR7ALDH1A1
SCHEMBL15113487 0.72 CHRM2 (0.30)
SCHEMBL1709238 0.72 SCN9A (0.59) SCN9ASIGMAR1HTR7ALDH1A1NPY1R
SCHEMBL1709236 0.71 SCN9A (1.00) SCN9ASIGMAR1DRD2USP2CYP2D6
SCHEMBL1709210 0.71 HTR1A (0.62) SCN9ASIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed