SCHEMBL1709237

SCHEMBL1709237

c1ccc(CCCNCC2CC23CCN(c2ccccc2)CC3)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.58
SIGMAR1 Q99720 8/20 0.45
HTR2A P28223 2/20 0.43
HRH1 P35367 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10071959 0.82 CCR3 (0.51) SCN9ASMN1; SMN2
SCHEMBL10071960 0.80 SCN9A (0.49) SCN9ANAMPT
SCHEMBL1709243 0.75 SCN9A (0.52) SCN9AHTR2A
SCHEMBL1709210 0.73 HTR1A (0.62) SCN9ASIGMAR1HTR1ADRD2NAMPT
SCHEMBL1709236 0.73 SCN9A (1.00) SCN9ASIGMAR1SMN1; SMN2HTR1ADRD2
SCHEMBL1709217 0.71 SCN9A (0.48) SCN9AHTR2A
SCHEMBL10072038 0.71 SCN9A (0.53) SCN9A
SCHEMBL1709249 0.70 DRD4 (0.60) SCN9ASIGMAR1HTR2AHTR1ADRD2
SCHEMBL1709241 0.70 SCN9A (0.54) SCN9ASIGMAR1DRD2
SCHEMBL1709252 0.69 SCN9A (0.56) SCN9ASIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed