SCHEMBL1011053

SCHEMBL1011053

Nc1ccccc1C(=O)Nc1ccc(Br)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.70
RAB9A P51151 1/20 0.70
PTGS1 P23219 3/20 0.65
FADS1 O60427 3/20 0.59
P2RX1 P51575 1/20 0.55
MAOB P27338 2/20 0.53
MAOA P21397 1/20 0.53
TP53 P04637 1/20 0.53
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
ALDH1A1 P00352 3/20 0.52
MAPT P10636 3/20 0.52
TDP1 Q9NUW8 1/20 0.51
LMNA P02545 2/20 0.51
HTT P42858 2/20 0.51
EGFR P00533 1/20 0.51
ERBB2 P04626 1/20 0.51
CYP1A2 P05177 1/20 0.51
LCK P06239 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30339241 1.00 NPC1 (0.70) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL17744848 0.91 PTGS1 (0.75) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL27826357 0.87 NPC1 (0.61) NPC1RAB9APTGS1FADS1MAOB
SCHEMBL30830441 0.86 PTGS1 (0.69) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL2127535 0.86 PTGS1 (0.69) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL1140055 0.85 PTGS1 (0.68) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL4954215 0.84 PTGS1 (0.67) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL4957349 0.84 LMNA (0.69) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL1961988 0.83 FADS1 (0.73) NPC1RAB9APTGS1FADS1P2RX1
SCHEMBL5925259 0.83 MAPT (0.59) NPC1RAB9APTGS1FADS1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240066136-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI), INC. (CN) 2024-02-29 US disclosed
CN-117510415-A Synthesis method of quinazolinone compound 中国人民解放军军事科学院防化研究院 2024-02-06 CN disclosed
CN-116472292-A Modified proteins and protein degrading agents 上海睿跃生物科技有限公司 2023-07-21 CN disclosed
US-20230057177-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI), INC. (CN) 2023-02-23 US disclosed
WO-2021239117-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI) , INC. (CN) 2021-12-02 WO disclosed
EP-2660238-B1 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP (CA) 2015-05-06 EP disclosed
EP-2660238-B1 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP (CA) 2015-05-06 EP disclosed
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US disclosed
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US disclosed
EP-2382194-B1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP (CA) 2014-03-12 EP disclosed
WO-2010079431-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2010-07-15 WO disclosed
WO-2010079431-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2010-07-15 WO disclosed
EP-1014962-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2007-06-27 EP disclosed
US-7067543-B2 Anthranilic acid amides and pharmaceutical use thereof NOVARTIS AG (CH) 2006-06-27 US disclosed
US-20040248947-A1 Anthranilic acid amides and pharmaceutical use thereof NOVARTIS AG (CH) 2004-12-09 US disclosed
US-6605626-B2 Benzamide inhibitors of factor Xa ELI LILLY AND COMPANY 2003-08-12 US disclosed
US-20020120007-A1 Benzamide inhibitors of factor Xa BEIGHT DOUGLAS WADE (US) 2002-08-29 US disclosed
US-6313122-B1 AS INHIBITORS OF FACTOR XA AND ARE USED AS ANTICOAGULANTS IN MAMMALS ELI LILLY AND COMPANY 2001-11-06 US disclosed
EP-1014962-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1999000121-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248947-A1 Anthranilic acid amides and pharmaceutical use thereof AFF1, FFAR1, FFAR2 NPC1 1201/4885RAB9A 1291/4885PTGS1 1909/4885
US-20240066136-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS DDB1, DCLRE1A, MDM2 NPC1 3949/4885RAB9A 3280/4885PTGS1 3614/4885
US-20020120007-A1 Benzamide inhibitors of factor Xa TFPI, F11, F12 NPC1 1618/4885RAB9A 2658/4885PTGS1 1623/4885
US-20230057177-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS DDB1, DCLRE1A, MDM2 NPC1 3949/4885RAB9A 3280/4885PTGS1 3614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.