SCHEMBL10123564

SCHEMBL10123564

Fc1cc2ccccn2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.48
NPC1 O15118 5/20 0.47
RAB9A P51151 5/20 0.47
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
POLB P06746 3/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
CHRNA7 P36544 1/20 0.34
HRH3 Q9Y5N1 3/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
NAMPT P43490 1/20 0.33
SSTR4 P31391 1/20 0.33
TP53 P04637 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3894978 0.78 ALDH1A1 (0.62) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL3895951 0.75 ALDH1A1 (0.58) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL24097278 0.74 ALOX15 (0.50) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL3896087 0.73 ALDH1A1 (0.47) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL321553 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL21824311 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL9517185 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL277387 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL2010683 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL15683854 0.73 ALOX15 (0.48) ALOX15NPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113563328-B Preparation method of 1, 3-disubstituted-2-fluoro indolizine derivative 台州学院 2022-07-05 CN disclosed
CN-113563328-B Preparation method of 1, 3-disubstituted-2-fluoro indolizine derivative 台州学院 2022-07-05 CN disclosed
CN-113563328-A Preparation method of 1, 3-disubstituted-2-fluoro indolizine derivative 台州学院 2021-10-29 CN disclosed
CN-113563328-A Preparation method of 1, 3-disubstituted-2-fluoro indolizine derivative 台州学院 2021-10-29 CN disclosed
WO-2014092478-A1 ORGANIC COMPOUND, AND ORGANIC ELECTROLUMINESCENCE DEVICE COMPRISING SAME 주식회사 두산 (KR) 2014-06-19 WO disclosed
US-8748452-B2 Indolizine derivative and use thereof for medical purposes KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-06-10 US disclosed
US-20120015972-A1 INDOLIZINE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES KISSEI PHARMACEUTICAL CO., LTD. (JP) 2012-01-19 US disclosed
US-20120015972-A1 INDOLIZINE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES KISSEI PHARMACEUTICAL CO., LTD. (JP) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015972-A1 INDOLIZINE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES XDH, INMT, PON1 ALOX15 467/4885NPC1 567/4885RAB9A 3005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.