SCHEMBL10146004

SCHEMBL10146004

Cc1ccc(Cn2c(=O)n(C)c3cc(-c4ccccc4N)ccc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.48
PARG Q86W56 2/20 0.47
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
GRM2 Q14416 1/20 0.44
PIK3CD O00329 1/20 0.43
GAA P10253 1/20 0.43
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
P2RX4 Q99571 1/20 0.41
HDAC1 Q13547 1/20 0.41
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HPD P32754 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14992138 0.83 PPARG (0.47) BRD4PARGMEN1KMT2AGRM2
SCHEMBL10145948 0.82 GRM2 (0.49) GRM2HPD
SCHEMBL10146668 0.80 GRM2 (0.70) PARGGRM2
SCHEMBL10145941 0.80 GRM2 (0.47) MEN1KMT2AGRM2ALDH1A1NPC1
SCHEMBL10146676 0.80 GRM2 (0.47) BRD4PARGGRM2ALDH1A1HPD
SCHEMBL10145950 0.79 MAPK14 (0.53) BRD4GRM2ALDH1A1KDM4EMAPT
SCHEMBL10145952 0.78 GRM2 (0.45) GRM2HDAC1NPC1KDM4EMAPT
SCHEMBL10146671 0.77 PARG (0.51) PARGGRM2
SCHEMBL10145910 0.73 GRM2 (0.60) PARGGRM2
SCHEMBL10145993 0.73 GRM2 (0.60) PARGGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed