SCHEMBL10175439

SCHEMBL10175439

Cn1cc(-c2cncc(-c3nc4cc(C#N)ccc4n3C)c2)cn1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.46
CSNK1A1 P48729 1/20 0.45
CSNK1D P48730 1/20 0.45
CSNK1G2 P78368 1/20 0.45
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
KCNJ5 P48544 1/20 0.40
KCNJ3 P48549 1/20 0.40
CYP11B1 P15538 4/20 0.39
FLT3 P36888 2/20 0.39
ATM Q13315 1/20 0.37
CCNK O75909 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
CDK12 Q9NYV4 1/20 0.37
MET P08581 1/20 0.36
LRRK2 Q5S007 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175123 0.87 CYP11B2 (0.64) CYP11B2CYP11B1
SCHEMBL10175348 0.83 CYP11B2 (0.48) CYP11B2CYP11B1ATM
SCHEMBL10175342 0.81 CYP11B2 (0.46) CYP11B2CYP11B1ATM
SCHEMBL17896641 0.81 CYP11B2 (0.47) CYP11B2CYP11B1ATM
SCHEMBL17896630 0.80 NPBWR1 (0.48) CYP11B2MKNK1MKNK2CYP11B1MET
SCHEMBL17896642 0.79 ALOX5AP (0.46) CYP11B2CYP11B1
SCHEMBL17883795 0.78 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL4243953 0.77 CYP11B2 (0.69) CYP11B2CYP11B1ATM
SCHEMBL10175442 0.77 BRD4 (0.46) CYP11B2CYP11B1
SCHEMBL10175456 0.76 MEN1 (0.57) CYP11B2CYP11B1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed