SCHEMBL10175616

SCHEMBL10175616

CC(C)n1c(-c2cncc(F)c2)nc2cc(NS(C)(=O)=O)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
USP2 O75604 2/20 0.42
HTT P42858 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
DYRK1A Q13627 1/20 0.41
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39
APLNR P35414 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MET P08581 4/20 0.38
CYP19A1 P11511 1/20 0.38
ADRA2B P18089 1/20 0.38
NR3C1 P04150 1/20 0.38
AR P10275 1/20 0.38
BRPF1 P55201 1/20 0.36
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896755 0.86 SMN1; SMN2 (0.44) CYP11B1CYP11B2DYRK1AALDH1A1POLB
SCHEMBL17883790 0.84 USP2 (0.63) CYP11B1CYP11B2USP2HTTNCOA1
SCHEMBL17883783 0.83 CYP11B2 (0.43) CYP11B1CYP11B2HTTDYRK1AALDH1A1
SCHEMBL10175462 0.81 KDM4E (0.42) CYP11B1CYP11B2HTTDYRK1AALDH1A1
SCHEMBL17896681 0.75 CYP11B2 (0.59) CYP11B1CYP11B2USP2HTTNCOA1
SCHEMBL17896587 0.74 CYP11B2 (0.73) CYP11B1CYP11B2USP2HTTNCOA1
SCHEMBL10175614 0.73 SMN1; SMN2 (0.46) DYRK1AALDH1A1POLBMETBRPF1
SCHEMBL17896756 0.71 PTGS2 (0.45) CYP11B1CYP11B2ALDH1A1POLBKDM4E
SCHEMBL460529 0.69 NAMPT (0.53) CYP11B1CYP11B2ALDH1A1METBRPF1
SCHEMBL10175126 0.68 CA12 (0.53) CYP11B1CYP11B2CYP19A1ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US claimed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed