SCHEMBL10177256

SCHEMBL10177256

OCn1cc(C(F)(F)F)nc1-c1ccc(Br)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.42
PTGS2 P35354 10/20 0.35
PTGS1 P23219 4/20 0.34
DGAT1 O75907 1/20 0.34
RXRA P19793 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
PDE2A O00408 2/20 0.32
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
APOBEC3A P31941 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
NOTUM Q6P988 2/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10177499 0.85 PTGS2 (0.35) PTGS2PTGS1RXRANR1H2NR1H3
SCHEMBL25975294 0.80 NT5E (0.44) NT5EPTGS2PTGS1RXRANR1H2
SCHEMBL9940375 0.79 DGAT1 (0.61) NT5EPTGS2PTGS1DGAT1RXRA
SCHEMBL10176917 0.79 DGAT1 (0.35) NT5EPTGS2PTGS1DGAT1ALDH1A1
SCHEMBL24185626 0.78 DGAT1 (0.45) PTGS2PTGS1DGAT1ALDH1A1
SCHEMBL20169324 0.78 DGAT1 (0.45) NT5EPTGS2PTGS1DGAT1RXRA
SCHEMBL10176667 0.74 PTGS2 (0.37) PTGS2PTGS1DGAT1
SCHEMBL25298735 0.74 USP1 (0.39) NT5EPTGS2PTGS1DGAT1
SCHEMBL25792027 0.73 PTGS2 (0.37) PTGS2PTGS1DGAT1RXRANR1H2
SCHEMBL30320360 0.73 PTGS2 (0.37) PTGS2PTGS1DGAT1RXRANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012081736-A1 CONTINUOUS ARYCYCLIC COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-06-21 WO disclosed