SCHEMBL1017772

SCHEMBL1017772

O=C(O)c1ccc(S(=O)(=O)CCc2ncc[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
TBXAS1 P24557 2/20 0.46
HSD17B10 Q99714 2/20 0.44
TSHR P16473 1/20 0.44
CA12 O43570 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
CA1 P00915 3/20 0.40
CA14 Q9ULX7 2/20 0.40
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CYP2C19 P33261 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
RAB9A P51151 1/20 0.39
SLC22A6 Q4U2R8 1/20 0.39
SLC22A8 Q8TCC7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5681941 0.79 TBXAS1 (0.55) ALDH1A1KDM4ETBXAS1KMT2ANAMPT
Hydrochloric Acid SCHEMBL8801622 0.78 ALDH1A1 (0.51) ALDH1A1KDM4ETBXAS1SMN1; SMN2LMNA
SCHEMBL7804458 0.75 PKM (0.53) ALDH1A1KDM4ETBXAS1HSD17B10TSHR
Hydrochloric Acid SCHEMBL9853948 0.73 TAAR1 (0.62) ALDH1A1KDM4ETBXAS1TSHRSMN1; SMN2
SCHEMBL4016565 0.71 TBXAS1 (0.50) TBXAS1SMN1; SMN2GAANAMPTTAAR1
SCHEMBL1018318 0.71 CA2 (0.60) ALDH1A1HSD17B10TSHRCA12CA2
SCHEMBL7869978 0.70 HTT (0.62) ALDH1A1KDM4EHSD17B10TSHRCA12
SCHEMBL1018690 0.70 CA12 (0.57) ALDH1A1HSD17B10TSHRCA12CA2
SCHEMBL2916604 0.70 TSHR (0.56) ALDH1A1HSD17B10TSHRCA12CA2
SCHEMBL1206780 0.70 MEP1B (0.50) ALDH1A1KDM4ETBXAS1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271642-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING Genentech, Inc. (US) 2011-01-12 EP disclosed
WO-2009126863-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING GENENTECH, INC. (US) 2009-10-15 WO disclosed
EP-1789390-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING Genentech, Inc. (US) 2007-05-30 EP disclosed
WO-2006028958-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING GENENTECH, INC. (US) 2006-03-16 WO disclosed