SCHEMBL10207451

SCHEMBL10207451

CON(C)C(=O)C1CCC(C(=O)c2ccc(Cl)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 11/20 0.50
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PKM P14618 1/20 0.44
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16309650 1.00 MGLL (0.50) MGLLLMNATP53MAPTL3MBTL1
SCHEMBL12292229 0.86 MGLL (0.48) MGLLLMNATP53MAPTL3MBTL1
SCHEMBL10207453 0.82 HSD17B1 (0.59) LMNATP53MAPTRAB9ANPC1
(4-Chlorophenyl)(Cyclopropyl)Methanone SCHEMBL392801 0.80 MGLL (0.68) MGLLLMNATP53MAPTL3MBTL1
SCHEMBL16762004 0.80 HSD17B1 (0.43) MAPTRAB9APKM
SCHEMBL16762006 0.80 HSD17B1 (0.43) MAPTRAB9APKM
SCHEMBL20683528 0.78 PKM (0.40) RAB9APKM
SCHEMBL12292711 0.78 HSD17B1 (0.41) LMNARAB9AMEN1KMT2APKM
SCHEMBL918622 0.77 NOTUM (0.54) LMNAMAPTRAB9AMEN1KMT2A
(4-Chlorophenyl)(Cyclopropyl)Methanone SCHEMBL6220062 0.77 MGLL (0.64) MGLLLMNATP53MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9994594-B2 Inhibitors of arginase and their therapeutic applications MARS, INCORPORATED (US) 2018-06-12 US disclosed
US-9994594-B2 Inhibitors of arginase and their therapeutic applications MARS, INCORPORATED (US) 2018-06-12 US disclosed
US-20170183362-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2017-06-29 US disclosed
US-9040703-B2 Inhibitors of arginase and their therapeutic applications MARS, INCORPORATED (US) 2015-05-26 US disclosed
US-20140371175-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2014-12-18 US disclosed
US-20120083469-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2012-04-05 US disclosed
US-20120083469-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170183362-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 MGLL 1073/4885LMNA 3157/4885TP53 3771/4885
US-20120083469-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 MGLL 1073/4885LMNA 3157/4885TP53 3771/4885
US-20140371175-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 MGLL 1073/4885LMNA 3157/4885TP53 3771/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.