SCHEMBL254376

SCHEMBL254376

COC(=O)[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(C)(C)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ESRRG P62508 1/20 0.40
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
EPHX2 P34913 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
APEX1 P27695 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
CYP26A1 O43174 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255310 0.87 NPC1 (0.38) CA2NPC1RAB9AESRRGADRB2
SCHEMBL254947 0.86 NPC1 (0.40) CA2NPC1RAB9AESRRGADRB2
SCHEMBL15235729 0.86 CA2 (0.39) CA2NPC1RAB9AESRRGADRB2
SCHEMBL255220 0.83 NPC1 (0.41) CA2NPC1RAB9AESRRG
SCHEMBL254164 0.81 NPC1 (0.36) CA2NPC1RAB9AESRRGADRB2
SCHEMBL1761476 0.80 TAS1R3 (0.59) CA2NPC1RAB9AMEN1LMNA
SCHEMBL254640 0.77 ACACB (0.41) CA2NPC1RAB9AESRRGADRB2
SCHEMBL20299901 0.77 ACACB (0.41) CA2NPC1RAB9AESRRGADRB2
SCHEMBL255440 0.76 TAS1R3 (0.48) CA2NPC1RAB9AADRB2ADRB1
SCHEMBL255181 0.76 TAS1R3 (0.48) CA2NPC1RAB9AADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed