SCHEMBL10272986

SCHEMBL10272986

CCc1cc(Cl)c(Cl)cn1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
ALDH1A1 P00352 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31651921 0.82 GRIN2D (0.38) CYP1A2POLBPTGS1PTGS2ALDH1A1
SCHEMBL10271475 0.82 NOS3 (0.35) CYP1A2POLBPTGS1PTGS2ALDH1A1
SCHEMBL20288204 0.82 NOS3 (0.35) CYP1A2POLBPTGS1PTGS2ALDH1A1
SCHEMBL12963743 0.80 GAA (0.35) GAAHTTCYP1A2POLBPTGS1
SCHEMBL25801524 0.80 GABRA1 (0.34) HTTCYP1A2POLBPTGS1PTGS2
SCHEMBL21262457 0.80 GAA (0.39) GAACYP1A2POLBPTGS1PTGS2
SCHEMBL16502348 0.80 PGK1 (0.37) CYP1A2POLBPTGS1PTGS2
SCHEMBL31652113 0.80 ALDH1A1 (0.32) CYP1A2POLBPTGS1PTGS2ALDH1A1
SCHEMBL14114852 0.79 PDXK (0.36) CYP1A2POLBPTGS1PTGS2ALDH1A1
SCHEMBL20642297 0.77 LMNA (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160101104-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL MYERS SQUIBB CO (US) 2016-04-14 US disclosed
US-20150342935-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL MYERS SQUIBB CO (US) 2015-12-03 US disclosed
US-20120035189-A1 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands BRISTOL-MYERS SQUIBB COMPANY 2012-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120035189-A1 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands CHRNA7, CHRNA5, CHRNA6 GAA 446/4885HTT 714/4885CYP1A2 2027/4885
US-20160101104-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA7, CHRNA5, CHRNA6 GAA 446/4885HTT 714/4885CYP1A2 2027/4885
US-20150342935-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA7, CHRNA5, CHRNA6 GAA 446/4885HTT 714/4885CYP1A2 2027/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.