SCHEMBL10285603

SCHEMBL10285603

C[C@@H]1CN(Cc2cc(Nc3nc4cccnc4s3)nc(Cl)n2)C[C@H](C)O1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.45
LCK P06239 1/20 0.45
AURKB Q96GD4 1/20 0.45
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.40
LMNA P02545 2/20 0.39
GAA P10253 1/20 0.39
RORC P51449 1/20 0.39
DHODH Q02127 1/20 0.39
ALK Q9UM73 1/20 0.38
KDM4E B2RXH2 4/20 0.38
HSD17B10 Q99714 1/20 0.38
SSTR5 P35346 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
HCRTR1 O43613 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL141353 0.82 ITK (0.68) ITKLCKAURKBRORCDHODH
SCHEMBL141352 0.82 ITK (0.68) ITKLCKAURKBRORCDHODH
SCHEMBL807713 0.78 ITK (0.41) ITKLCKAURKBNPC1POLB
SCHEMBL2395616 0.77 ITK (0.56) ITKLCKAURKBPOLBRORC
SCHEMBL807540 0.75 ITK (0.46) ITKLCKAURKBNPC1RAB9A
SCHEMBL807946 0.71 ITK (0.58) ITKLCKAURKBRORCDHODH
SCHEMBL808093 0.71 ITK (0.61) ITKLCKAURKBRORCDHODH
SCHEMBL807743 0.71 ITK (0.57) ITKLCKAURKBRORCDHODH
SCHEMBL807803 0.70 ITK (0.58) ITKLCKAURKBRORCDHODH
SCHEMBL807804 0.70 LCK (0.46) ITKLCKAURKBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed