SCHEMBL808093

SCHEMBL808093

C/C=C/C(=O)N1CC[C@H](Nc2cc(CN3C[C@@H](C)O[C@@H](C)C3)cc(Nc3nc4cccnc4s3)n2)C1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.61
RORC P51449 1/20 0.42
DHODH Q02127 1/20 0.42
BTK Q06187 11/20 0.41
HCK P08631 9/20 0.41
SSTR5 P35346 1/20 0.40
LCK P06239 1/20 0.39
AURKB Q96GD4 1/20 0.39
LTA4H P09960 1/20 0.33
JAK3 P52333 3/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285825 0.92 ITK (0.58) ITKRORCDHODHBTKHCK
SCHEMBL807743 0.90 ITK (0.57) ITKRORCDHODHBTKHCK
SCHEMBL807946 0.88 ITK (0.58) ITKRORCDHODHBTKHCK
SCHEMBL807803 0.87 ITK (0.58) ITKRORCDHODHBTKHCK
SCHEMBL808081 0.84 ITK (0.54) ITKRORCDHODHBTKHCK
SCHEMBL2395616 0.83 ITK (0.56) ITKRORCDHODHBTKSSTR5
SCHEMBL808096 0.83 ITK (0.51) ITKRORCDHODHBTKHCK
SCHEMBL22374670 0.83 ITK (0.71) ITKRORCDHODHBTKHCK
SCHEMBL807540 0.80 ITK (0.46) ITKRORCDHODHSSTR5LCK
SCHEMBL807926 0.78 ITK (0.59) ITKRORCDHODHBTKHCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed