SCHEMBL807743

SCHEMBL807743

C/C=C(\C)C(=O)N1CC[C@H](Nc2cc(CN3C[C@@H](C)O[C@@H](C)C3)cc(Nc3nc4cccnc4s3)n2)C1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.57
RORC P51449 1/20 0.42
DHODH Q02127 1/20 0.42
SSTR5 P35346 1/20 0.40
LCK P06239 1/20 0.39
AURKB Q96GD4 1/20 0.39
BTK Q06187 10/20 0.38
HCK P08631 8/20 0.38
KDR P35968 2/20 0.34
MLNR O43193 2/20 0.33
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807946 0.92 ITK (0.58) ITKRORCDHODHSSTR5LCK
SCHEMBL808093 0.90 ITK (0.61) ITKRORCDHODHSSTR5LCK
SCHEMBL807803 0.87 ITK (0.58) ITKRORCDHODHSSTR5LCK
SCHEMBL808081 0.87 ITK (0.54) ITKRORCDHODHSSTR5LCK
SCHEMBL10285825 0.86 ITK (0.58) ITKRORCDHODHSSTR5LCK
SCHEMBL2395616 0.83 ITK (0.56) ITKRORCDHODHSSTR5LCK
SCHEMBL808096 0.83 ITK (0.51) ITKRORCDHODHSSTR5LCK
SCHEMBL807540 0.80 ITK (0.46) ITKRORCDHODHSSTR5LCK
SCHEMBL22374670 0.80 ITK (0.71) ITKRORCDHODHSSTR5LCK
SCHEMBL807926 0.78 ITK (0.59) ITKRORCDHODHSSTR5LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed