SCHEMBL10287802

SCHEMBL10287802

CN1CC(c2ccccc2)C=N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
BRD4 O60885 3/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
SRD5A1 P18405 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
DRD5 P21918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14275214 0.74 MAPT (0.34) ALDH1A1CHRNA7KMT2A
SCHEMBL1843873 0.70 MAOB (0.39) ALDH1A1MAOAMAOBKMT2A
SCHEMBL4486104 0.70 HTR6 (0.33)
SCHEMBL30009253 0.69 MAOB (0.40) ALDH1A1MAOAMAOB
SCHEMBL30630035 0.69 MAOA (0.34) MAOAMAOBSLC6A2HTR1A
SCHEMBL13791492 0.69 CYP2A6 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30009763 0.69 RIPK1 (0.36) ALDH1A1HPGDMAOAMAOBSLC6A3
Hydrochloric Acid SCHEMBL31478169 0.68 RIPK1 (0.35) ALDH1A1HPGDMAOAMAOBKMT2A
SCHEMBL12671459 0.66
SCHEMBL14870536 0.64 CHRNB2 (0.59) ALDH1A1BRD4CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037411-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
CN-101137377-A Tetracyclic amino and carboxamido compounds and methods of use thereof INOTEK PHARMACEUTICALS CORP (US) 2008-03-05 CN disclosed
CN-1170434-A In vitro Induction of dopaminergic cells NEUROSPHERES HOLDINGS LTD (US) 1998-01-14 CN disclosed
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed