SCHEMBL10301957

SCHEMBL10301957

C=CCOc1ccc(-c2ccc(CCc3ccc(C)c(F)c3F)cc2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.35
HTR2C P28335 6/20 0.34
HTR2B P41595 4/20 0.34
S1PR1 P21453 1/20 0.33
ERN1 O75460 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
HTR2A P28223 2/20 0.31
LMNA P02545 1/20 0.31
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP2D6 P10635 1/20 0.31
PTGER2 P43116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10301958 0.89 S1PR1 (0.36) CYP17A1S1PR1MAPT
SCHEMBL10301959 0.88 S1PR1 (0.37) CYP17A1S1PR1MAPT
SCHEMBL12735665 0.87 FFAR4 (0.36) CYP17A1HTR2CHTR2BS1PR1ERN1
SCHEMBL10301952 0.86 NAAA (0.40) CYP17A1S1PR1ALDH1A1KDM4EMAPT
SCHEMBL10301931 0.84 CTSS (0.37) HTR2CHTR2BALDH1A1KDM4EMAPT
SCHEMBL10302482 0.84 FFAR1 (0.36) HTR2CHTR2BERN1
SCHEMBL10302989 0.84 LMNA (0.35) CYP17A1HTR2CHTR2BS1PR1ERN1
SCHEMBL10302227 0.84 ERN1 (0.42) CYP17A1HTR2CHTR2BERN1ALDH1A1
SCHEMBL12738911 0.84 PTGS2 (0.34) CYP17A1HTR2CHTR2BS1PR1ERN1
SCHEMBL10301953 0.83 S1PR1 (0.48) CYP17A1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8216489-B2 Three-ring liquid crystal compound having lateral fluorine, liquid crystal composition, and liquid crystal display device JNC CORPORATION (JP) 2012-07-10 US disclosed
US-20110037024-A1 THREE-RING LIQUID CRYSTAL COMPOUND HAVING LATERAL FLUORINE, LIQUID CRYSTAL COMPOSITION, AND LIQUID CRYSTAL DISPLAY DEVICE CHISSO CORPORATION (JP) 2011-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110037024-A1 THREE-RING LIQUID CRYSTAL COMPOUND HAVING LATERAL FLUORINE, LIQUID CRYSTAL COMPOSITION, AND LIQUID CRYSTAL DISPLAY DEVICE LEF1, LAS1L, L3MBTL3 CYP17A1 1641/4885HTR2C 770/4885HTR2B 1904/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.