SCHEMBL1030480

SCHEMBL1030480

COc1cccc(CN(CC2CCCO2)C(=O)c2c(-c3ccco3)c(C)cn2C)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
GAA P10253 3/20 0.46
POLB P06746 2/20 0.46
TP53 P04637 1/20 0.46
LMNA P02545 3/20 0.46
HSD17B10 Q99714 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
OXTR P30559 4/20 0.44
AVPR1A P37288 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
TSHR P16473 2/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
MAPT P10636 1/20 0.42
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1032230 0.74 ADORA3 (0.55) ALDH1A1POLBTP53LMNAKDM4E
SCHEMBL1032179 0.69 ADORA3 (0.49) ALDH1A1POLBTP53LMNAKDM4E
SCHEMBL5808402 0.68 ALDH1A1 (0.61) ALDH1A1GAAPOLBTP53LMNA
SCHEMBL5808404 0.68 ALDH1A1 (0.61) ALDH1A1GAAPOLBTP53LMNA
SCHEMBL5808248 0.67 ALDH1A1 (0.54) ALDH1A1GAAPOLBTP53HSD17B10
SCHEMBL20387961 0.64 ALDH1A1 (0.78) ALDH1A1GAAPOLBLMNAKDM4E
SCHEMBL1030274 0.64 POLB (0.46) ALDH1A1GAAPOLBLMNAHSD17B10
SCHEMBL1031744 0.63 NPC1 (0.49) ALDH1A1POLBLMNAHSD17B10KDM4E
SCHEMBL1031849 0.63 ALDH1A1 (0.49) ALDH1A1GAAPOLBTP53LMNA
SCHEMBL9416588 0.62 HSD17B2 (0.57) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed