SCHEMBL5808248

SCHEMBL5808248

COc1cccc(CN(CC2CCCO2)C(=O)c2cccc(C=C[Si](O)(O)C(C)C)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
GAA P10253 4/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 3/20 0.49
POLB P06746 2/20 0.49
MEN1 O00255 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
OXTR P30559 5/20 0.47
AVPR1A P37288 5/20 0.47
WDR5 P61964 1/20 0.44
NPC1 O15118 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5808404 0.70 ALDH1A1 (0.61) ALDH1A1GAATP53HPGDPOLB
SCHEMBL5804466 0.70 KMT2A (0.46) ALDH1A1MEN1TSHRKMT2A
SCHEMBL5805616 0.69 TRPM8 (0.50) TSHROXTR
SCHEMBL5808402 0.68 ALDH1A1 (0.61) ALDH1A1GAATP53HPGDPOLB
SCHEMBL1030480 0.67 ALDH1A1 (0.54) ALDH1A1GAATP53HPGDPOLB
SCHEMBL5806073 0.66 NR1H4 (0.44) ALDH1A1HPGDMEN1MAPK1KMT2A
SCHEMBL5804372 0.63 TP53 (0.55) ALDH1A1GAATP53MEN1ALOX15
SCHEMBL5804375 0.63 TP53 (0.55) ALDH1A1GAATP53MEN1ALOX15
SCHEMBL29171443 0.63 HPGD (0.60) ALDH1A1GAAHPGDPOLBMEN1
SCHEMBL25414340 0.63 OXTR (0.56) ALDH1A1HPGDPOLBMEN1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006069096-A1 SILANOL DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE PHARMACYCLICS, INC. (US) 2006-06-29 WO disclosed