SCHEMBL1030828

SCHEMBL1030828

Cc1ccc(C(=O)c2c(C)cn(Cc3ccc(F)cc3)c2C(=O)N2CCOCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.44
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
THRB P10828 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
MAPK1 P28482 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
EPHX2 P34913 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1029484 0.91 HSD11B1 (0.47) ALDH1A1THRBRXFP1
SCHEMBL1028758 0.84 GRIN2B (0.44) MAPTALDH1A1SMN1; SMN2MAPK1MEN1
SCHEMBL1031510 0.83 MEN1 (0.51) MEN1KMT2A
SCHEMBL1031811 0.82 HPGD (0.54) MAPTPOLBALDH1A1HPGDLMNA
SCHEMBL1034078 0.81 MAPT (0.46) MAPTPOLBGAAALDH1A1LMNA
SCHEMBL1028175 0.80 TP53 (0.52) MAPTPOLBALDH1A1LMNASMN1; SMN2
SCHEMBL1031573 0.79 KMT2A (0.52) MAPTALDH1A1LMNAMEN1KMT2A
SCHEMBL1030438 0.78 MEN1 (0.61) MAPTPOLBALDH1A1CYP2C19CYP2C9
SCHEMBL1032620 0.78 HTT (0.53) MAPTPOLBALDH1A1HPGDLMNA
SCHEMBL1029485 0.77 HSD11B1 (0.46) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed