SCHEMBL1029484

SCHEMBL1029484

Cc1ccc(C(=O)c2c(C)cn(Cc3ccc(F)cc3)c2C(=O)N2CCN(C(=O)c3ccc(C)cc3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.47
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
THRB P10828 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030828 0.91 MAPT (0.47) ALDH1A1THRBRXFP1
SCHEMBL1031510 0.88 MEN1 (0.51)
SCHEMBL1029485 0.86 HSD11B1 (0.46) HSD11B1ALDH1A1PKMCA12CA1
SCHEMBL1034078 0.86 MAPT (0.46) ALDH1A1
SCHEMBL1031811 0.84 HPGD (0.54) ALDH1A1PKM
SCHEMBL1028175 0.83 TP53 (0.52) ALDH1A1PKM
SCHEMBL1030438 0.82 MEN1 (0.61) ALDH1A1PKMTHRBL3MBTL1
SCHEMBL1032620 0.82 HTT (0.53) ALDH1A1
SCHEMBL1031573 0.82 KMT2A (0.52) HSD11B1ALDH1A1
SCHEMBL1032634 0.80 ALDH1A1 (0.41) ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed