SCHEMBL10312557

SCHEMBL10312557

Cc1ccc(-c2noc(CC(O[Si](C)(C)C(C)(C)C)C(=O)O[Si](C)(C)C(C)(C)C)n2)nc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 11/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
PSMB5 P28074 1/20 0.33
MAPT P10636 1/20 0.33
HDAC4 P56524 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548460 0.89 HCAR2 (0.36) HCAR2NPC1RAB9ASMN1; SMN2GAA
SCHEMBL10312561 0.76 HCAR2 (0.46) HCAR2NPC1RAB9ASMN1; SMN2GAA
SCHEMBL10312550 0.74 HCAR2 (0.51) HCAR2NPC1RAB9ASMN1; SMN2GAA
SCHEMBL10312560 0.72 CYP2C9 (0.46) HCAR2NPC1RAB9ASMN1; SMN2GAA
SCHEMBL10312554 0.72 RAB9A (0.49) HCAR2NPC1RAB9ASMN1; SMN2GAA
SCHEMBL10312532 0.69 MITF (0.54) HCAR2CYP2C9ALDH1A1TSHRMAPT
SCHEMBL10312533 0.69 MAPT (0.48) HCAR2SMN1; SMN2CYP2C9ALDH1A1TSHR
SCHEMBL13781597 0.68 TP53 (0.43) HCAR2NPC1RAB9ASMN1; SMN2CYP2C9
SCHEMBL10312563 0.68 TP53 (0.54) HCAR2RAB9ASMN1; SMN2GAACYP2C9
SCHEMBL11202582 0.67 SRR (0.43) MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178750-A1 Niacin Receptor Agonists, Compositions Containing Such Compounds and Methods of Treatment MERCK SHARP & DOHME CORP. (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178750-A1 Niacin Receptor Agonists, Compositions Containing Such Compounds and Methods of Treatment HCAR1, HCAR2, FFAR1 HCAR2 2/4885NPC1 19/4885RAB9A 2712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.