SCHEMBL1031909

SCHEMBL1031909

COc1ccc(OCCNC(=O)c2c(-c3ccccc3)c(C)cn2Cc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
RECQL P46063 1/20 0.47
ALDH1A1 P00352 3/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KMT2A Q03164 5/20 0.45
MEN1 O00255 1/20 0.45
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TSHR P16473 2/20 0.44
HPGD P15428 2/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FAAH O00519 1/20 0.42
ACHE P22303 1/20 0.42
BRD4 O60885 2/20 0.42
LMNA P02545 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1048091 0.81 ALDH1A1 (0.53) RAB9AALDH1A1SMN1; SMN2HPGDTP53
SCHEMBL1032474 0.78 NPC1 (0.44) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL1031481 0.78 THRB (0.53) NPC1RAB9AKMT2ASMN1; SMN2TP53
SCHEMBL1028264 0.76 CACNA1G (0.47) NPSR1KMT2AMEN1FAAHACHE
SCHEMBL1033446 0.76 NPC1 (0.53) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL1030734 0.76 CNR1 (0.45) NPC1ALDH1A1KMT2AMEN1HPGD
SCHEMBL1028724 0.74 POLB (0.51) NPC1RAB9AALDH1A1KMT2ASMN1; SMN2
SCHEMBL1033737 0.74 NPC1 (0.49) NPC1RAB9ARECQLALDH1A1KMT2A
SCHEMBL2638817 0.74 NOTUM (0.48) ALDH1A1SMN1; SMN2TSHRHPGDTP53
SCHEMBL1031690 0.74 HPGD (0.46) NPC1RAB9AALDH1A1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed