SCHEMBL10325542

SCHEMBL10325542

CCC(C(=O)O)C1CCN(c2ncc(-c3ccc(C=O)cn3)cn2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.37
AOC3 Q16853 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 3/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MITF O75030 1/20 0.35
KLF5 Q13887 1/20 0.35
HDAC3 O15379 3/20 0.34
HDAC4 P56524 3/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC7 Q8WUI4 3/20 0.34
HDAC2 Q92769 3/20 0.34
HDAC10 Q969S8 3/20 0.34
HDAC11 Q96DB2 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC9 Q9UKV0 3/20 0.34
HDAC5 Q9UQL6 3/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10325755 0.85 AOC3 (0.33) GPR119AOC3ALDH1A1KDM4EHDAC3
SCHEMBL10324413 0.81 DGAT1 (0.46) GPR119DGAT1
SCHEMBL10324422 0.69 DGAT1 (0.43) DGAT1
SCHEMBL1976988 0.67 AKR1C3 (0.46)
SCHEMBL4435638 0.67 ITGB3 (0.46)
SCHEMBL10379629 0.65 FFAR4 (0.37) GPR119AOC3KDM4EDGAT1
SCHEMBL25197619 0.65 AOC3 (0.42) GPR119AOC3KDM4EHDAC3HDAC4
SCHEMBL31584001 0.65 ALKBH1 (0.50)
SCHEMBL10324328 0.64 DGAT1 (0.56) DGAT1
SCHEMBL24409278 0.64 KDM5B (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed