SCHEMBL10324422

SCHEMBL10324422

CCC(C(=O)O)C1CCN(c2ccc(-c3ccc(C=O)c(F)c3)cn2)CC1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 13/20 0.43
KCNH2 Q12809 12/20 0.43
ADORA2A P29274 8/20 0.43
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
ERN1 O75460 1/20 0.39
MELK Q14680 3/20 0.39
SCD O00767 1/20 0.38
FFAR4 Q5NUL3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324875 0.89 MELK (0.40) MELKSCDFFAR4
SCHEMBL10326401 0.89 MELK (0.39) MELKFFAR4
SCHEMBL10380728 0.69 FFAR4 (0.43) DGAT1FFAR4
SCHEMBL10325542 0.69 GPR119 (0.37) DGAT1
SCHEMBL17729168 0.69 IDO1 (0.54)
SCHEMBL10380233 0.69 FFAR4 (0.41) DGAT1KCNH2ADORA2AFFAR4
SCHEMBL10379959 0.69 DGAT1 (0.47) DGAT1KCNH2ADORA2AERN1MELK
SCHEMBL10325123 0.66 KDM4E (0.46) MELK
SCHEMBL1727604 0.65 HTR1A (0.41) DGAT1KCNH2ADORA2ASCD
SCHEMBL14969291 0.64 ERN1 (0.46) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed