Xenbucin

Xenbucin

SCHEMBL10345475

CC(O)N(C)C.CCC(C(=O)O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.51
AKR1C3 P42330 4/20 0.46
AKR1C2 P52895 4/20 0.46
HTR1A P08908 1/20 0.46
ADRA1A P35348 1/20 0.46
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
ADAMTS4 O75173 1/20 0.43
KCNQ2 O43526 1/20 0.43
MAPT P10636 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
AKR1C1 Q04828 1/20 0.41
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xenbucin SCHEMBL24134 0.89 PTGS2 (0.58) PTGS2AKR1C3AKR1C2HTR1AADRA1A
Xenbucin SCHEMBL3360074 0.85 PTGS2 (0.55) PTGS2AKR1C3AKR1C2HTR1AADRA1A
Xenbucin SCHEMBL10345476 0.82 PTGS2 (0.45) PTGS2AKR1C3AKR1C2HTR1AADRA1A
SCHEMBL10345479 0.81 KCNQ2 (0.45) PTGS2AKR1C3AKR1C2HTR1AADRA1A
SCHEMBL1715 0.78 LMNA (0.59) HTR1AADRA1ACRHBPCRHR2KCNQ2
SCHEMBL67237 0.78 LMNA (0.59) HTR1AADRA1ACRHBPCRHR2KCNQ2
SCHEMBL65737 0.78 LMNA (0.59) HTR1AADRA1ACRHBPCRHR2KCNQ2
SCHEMBL29757088 0.78 LMNA (0.59) HTR1AADRA1ACRHBPCRHR2KCNQ2
SCHEMBL20769804 0.78 LMNA (0.59) HTR1AADRA1ACRHBPCRHR2KCNQ2
SCHEMBL1574429 0.78 AKR1C3 (0.58) PTGS2AKR1C3AKR1C2HTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0105635-B1 NONIRRITATING AQUEOUS OPHTHALMIC COMPOSITIONS COMFORT FORMULATION FOR OCULAR THEREPEUTIC AGENTS ALCON LABORATORIES, INC. (US) 1990-04-04 EP disclosed
US-4559343-A ANTIINFLAMMATORY AGENT WITH XANTHINE DERIVATIVE ALCON LABORATORIES, INC. (US) 1985-12-17 US disclosed
EP-0105635-A2 Nonirritating aqueous ophthalmic compositions comfort formulation for ocular therepeutic agents ALCON LABORATORIES, INC. (US) 1984-04-18 EP disclosed