Xenbucin

Xenbucin

SCHEMBL10345476

CCC(C(=O)O)c1ccc(-c2ccccc2)cc1.CN(C)CCO

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.45
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 2/20 0.44
KCNQ2 O43526 1/20 0.44
MAPT P10636 1/20 0.44
UTS2R Q9UKP6 9/20 0.43
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
UBE2N P61088 1/20 0.42
HTR1A P08908 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xenbucin SCHEMBL24134 0.86 PTGS2 (0.58) PTGS2AKR1C3AKR1C2KCNQ2MAPT
Xenbucin SCHEMBL3360074 0.83 PTGS2 (0.55) PTGS2AKR1C3AKR1C2KCNQ2MAPT
Xenbucin SCHEMBL10345475 0.82 PTGS2 (0.51) PTGS2AKR1C3AKR1C2KCNQ2MAPT
SCHEMBL10345478 0.79 CHRM1 (0.63) UTS2RKDM4EALDH1A1
SCHEMBL67237 0.76 LMNA (0.59) KCNQ2MAPTALDH1A1HTR1AADRA1A
SCHEMBL65737 0.76 LMNA (0.59) KCNQ2MAPTALDH1A1HTR1AADRA1A
SCHEMBL1715 0.76 LMNA (0.59) KCNQ2MAPTALDH1A1HTR1AADRA1A
SCHEMBL29757088 0.76 LMNA (0.59) KCNQ2MAPTALDH1A1HTR1AADRA1A
SCHEMBL20769804 0.76 LMNA (0.59) KCNQ2MAPTALDH1A1HTR1AADRA1A
SCHEMBL1574429 0.76 AKR1C3 (0.58) PTGS2AKR1C3AKR1C2ALDH1A1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0105635-B1 NONIRRITATING AQUEOUS OPHTHALMIC COMPOSITIONS COMFORT FORMULATION FOR OCULAR THEREPEUTIC AGENTS ALCON LABORATORIES, INC. (US) 1990-04-04 EP disclosed
US-4559343-A ANTIINFLAMMATORY AGENT WITH XANTHINE DERIVATIVE ALCON LABORATORIES, INC. (US) 1985-12-17 US disclosed
EP-0105635-A2 Nonirritating aqueous ophthalmic compositions comfort formulation for ocular therepeutic agents ALCON LABORATORIES, INC. (US) 1984-04-18 EP disclosed