SCHEMBL10366100

SCHEMBL10366100

N#Cc1c(C(=O)O)cnn1-c1ccc(Br)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NR4A3 Q92570 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
MAPK14 Q16539 3/20 0.39
MEN1 O00255 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963674 0.86 POLB (0.55) XDHSMN1; SMN2L3MBTL1NR4A3POLB
SCHEMBL2870416 0.85 PTPN1 (0.46) XDHSMN1; SMN2L3MBTL1NR4A3POLB
SCHEMBL10893230 0.85 MAPK14 (0.53) XDHSMN1; SMN2L3MBTL1NR4A3POLB
SCHEMBL10890676 0.85 RAB9A (0.49) XDHSMN1; SMN2L3MBTL1NR4A3POLB
SCHEMBL10892897 0.84 XDH (0.43) XDHSMN1; SMN2L3MBTL1NR4A3POLB
SCHEMBL10833122 0.83 ALDH1A1 (0.38) XDHSMN1; SMN2L3MBTL1KEAP1NFE2L2
SCHEMBL10365343 0.83 NPC1 (0.47) XDHSMN1; SMN2POLBMAPK14MEN1
SCHEMBL10896747 0.83 L3MBTL1 (0.44) SMN1; SMN2L3MBTL1NR4A3POLBMAPT
SCHEMBL10895563 0.82 PTPN1 (0.54) SMN1; SMN2MAPTMAPK14NPC1RAB9A
SCHEMBL10340580 0.81 ALDH1A1 (0.55) SMN1; SMN2MAPTMEN1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631343-A Cyanopyrazole intermediates ELI LILLY AND COMPANY (US) 1986-12-23 US claimed
EP-0151867-B1 CYANOPYRAZOLE HERBICIDES ELI LILLY AND COMPANY (US) 1990-01-10 EP disclosed
US-4631343-A Cyanopyrazole intermediates ELI LILLY AND COMPANY (US) 1986-12-23 US disclosed
US-4589905-A TERRESTRIAL AND AQUATIC APPLICATIONS ELI LILLY AND COMPANY (US) 1986-05-20 US disclosed
EP-0151867-A2 Cyanopyrazole herbicides ELI LILLY AND COMPANY (US) 1985-08-21 EP disclosed