SCHEMBL1037692

SCHEMBL1037692

C1=Cc2ccc3occc3c2NC1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
FTO Q9C0B1 1/20 0.32
NFKB1 P19838 1/20 0.31
CDK1 P06493 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
EED O75530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13791237 0.74
SCHEMBL14363754 0.70
SCHEMBL29474440 0.69 HTR2A (0.42) HTR2CHTR2AHTR2BMAOAMAOB
SCHEMBL8553982 0.67 CYP1A1 (0.40) HTR2CHTR2AHTR2BMAOAMAOB
SCHEMBL29657636 0.67 CYP1A1 (0.40) HTR2CHTR2AHTR2BMAOAMAOB
SCHEMBL14251852 0.66 MAOA (0.34) HTR2CHTR2AHTR2BMAOAMAOB
SCHEMBL5822842 0.66 HTR2C (0.33) HTR2C
SCHEMBL4429415 0.65 PAX8 (0.48) HTR2CHTR2AHTR2BMAOAMAOB
SCHEMBL70023 0.64 MAPT (0.48) NFKB1CDK1MAPKAPK2
SCHEMBL9411925 0.64 HTR2C (0.57) HTR2CHTR2AHTR2BMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250289830-A1 KRAS INHIBITORS ELI LILLY AND COMPANY 2025-09-18 US disclosed
US-12351591-B2 KRas inhibitors ELI LILLY AND COMPANY (US) 2025-07-08 US disclosed
EP-4499233-A1 KRAS INHIBITORS Eli Lilly and Company (US) 2025-02-05 EP disclosed
CN-119095853-A KRAS inhibitors 伊莱利利公司 2024-12-06 CN disclosed
US-20240043451-A1 KRAS INHIBITORS ELI LILLY AND COMPANY 2024-02-08 US disclosed
WO-2023183585-A1 KRAS INHIBITORS ELI LILLY AND COMPANY (US) 2023-09-28 WO disclosed
CN-110642866-B Dihydrofuranquinoline derivative and synthesis method and application thereof 广西师范大学 2021-08-03 CN disclosed
CN-110642866-A Dihydrofuranquinoline derivative and synthesis method and application thereof 广西师范大学 2020-01-03 CN disclosed
US-8012961-B2 Tricyclic antibiotics ACTELION PHARMACEUTICAL LTD. (CH) 2011-09-06 US disclosed
US-20110039836-A1 TRICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD. (CH) 2011-02-17 US disclosed
EP-2276766-A1 TRICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2011-01-26 EP disclosed
WO-2009128019-A1 TRICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2009-10-22 WO disclosed
EP-0063137-A1 STABILIZATION OF SUBSTITUTED 8-HYDROXYQUINOLINE HYDROMETALLURGICAL REAGENTS SHEREX CHEMICAL COMPANY, INC. (US) 1982-10-27 EP disclosed
WO-1982001369-A1 STABILIZATION OF SUBSTITUTED 8-HYDROXYQUINOLINE HYDROMETALLURGICAL REAGENTS SHEREX CHEM (US) 1982-04-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240043451-A1 KRAS INHIBITORS KRAS, NRAS, HRAS HTR2C 4816/4885HTR2A 4723/4885HTR2B 4592/4885
US-12351591-B2 KRas inhibitors KRAS, NRAS, HRAS HTR2C 4816/4885HTR2A 4723/4885HTR2B 4592/4885
US-20250289830-A1 KRAS INHIBITORS KRAS, NRAS, HRAS HTR2C 4816/4885HTR2A 4723/4885HTR2B 4592/4885
US-20110039836-A1 TRICYCLIC ANTIBIOTICS OPRM1, UBE2D3, METTL3 HTR2C 524/4885HTR2A 1310/4885HTR2B 2487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.