SCHEMBL10429353

SCHEMBL10429353

NC(=O)c1ccnc(-c2cccc(C(F)(F)F)c2)c1N

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
PARP1 P09874 2/20 0.53
KMO O15229 2/20 0.48
RORB Q92753 5/20 0.46
TDO2 P48775 1/20 0.45
KIF11 P52732 1/20 0.45
AURKA O14965 1/20 0.45
RPS6KB1 P23443 1/20 0.45
AURKB Q96GD4 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
RORC P51449 1/20 0.44
SYK P43405 1/20 0.44
JAK2 O60674 1/20 0.43
PDGFRB P09619 1/20 0.43
KDR P35968 1/20 0.43
GPR52 Q9Y2T5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5178386 0.84 PARP1 (0.58) KDM4EPARP1KMORORBKIF11
SCHEMBL1758364 0.78 IKBKB (0.47) KDM4EPARP1JAK2KDR
SCHEMBL8936345 0.76 KMO (0.54) KDM4EKMORORBTDO2ADORA2A
SCHEMBL9002267 0.75 RORB (0.56) PARP1KMORORBTDO2RORC
SCHEMBL34469502 0.75 KDM4E (0.51) KDM4EPARP1KMOKIF11AURKA
SCHEMBL11401523 0.75 PARP1 (0.51) KDM4EPARP1RORBKIF11ADORA2A
SCHEMBL34469496 0.75 PARP1 (0.54) KDM4EPARP1KMORORBKIF11
SCHEMBL10429369 0.74 GPR52 (0.45) KDM4ERORBGPR52
SCHEMBL4724483 0.74 PARP1 (0.59) KDM4EPARP1RORBKIF11ADORA1
SCHEMBL473595 0.74 ALDH1A1 (0.59) KDM4EPARP1KMORORBTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed