SCHEMBL8936345

SCHEMBL8936345

Nc1ccnc(-c2cccc(C(F)(F)F)c2)c1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.54
ADORA1 P30542 3/20 0.47
ADORA2A P29274 2/20 0.47
XDH P47989 1/20 0.46
HSD17B10 Q99714 2/20 0.46
HTT P42858 1/20 0.46
RORB Q92753 5/20 0.46
TDO2 P48775 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PIN1 Q13526 1/20 0.43
HPGD P15428 1/20 0.42
KCNA5 P22460 2/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CG P48736 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19138009 0.80 HTT (0.46) HSD17B10HTTKDM4EALDH1A1
SCHEMBL3345499 0.78 KMO (0.56) KMOADORA1ADORA2AXDHRORB
SCHEMBL8691066 0.77 TDO2 (0.46) KMOADORA1ADORA2AXDHRORB
SCHEMBL9048030 0.77 ADORA2A (0.48) KMOADORA1ADORA2ARORBTDO2
SCHEMBL368305 0.77 DHODH (0.47) HSD17B10HTT
SCHEMBL473595 0.77 ALDH1A1 (0.59) KMOXDHRORBTDO2KDM4E
SCHEMBL10429353 0.76 KDM4E (0.55) KMOADORA1ADORA2ARORBTDO2
SCHEMBL13734158 0.76 BRD4 (0.53) KMOADORA1ADORA2AXDHRORB
SCHEMBL9047986 0.76 ADORA2A (0.48) ADORA1ADORA2AXDHTDO2PIN1
SCHEMBL31606903 0.76 ADORA2A (0.51) ADORA1ADORA2AXDHTDO2KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996031469-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed
US-5541174-A COORDINATION COMPOUND OF COPPER AND AN AMINO ACID SORENSON JOHN R J (US) 1996-07-30 US disclosed
US-5216021-A Copper coordination compounds SORENSON JOHN R J (US) 1993-06-01 US disclosed
US-5082834-A Antiarthritic agents, coordination compounds of copper and aci d salicylates J.R.J. SORENSON CORP. 1992-01-21 US disclosed
US-4440754-A COPPER COORDINATION COMPOUNDS J.R.J. SORENSON CORP. 1984-04-03 US disclosed
US-4221785-A COORDINATION COMPOUND OF A COPPER SALT AND A SALICYLIC ACID OR ITS DERIVATIVE J.R.J. SORENSON CORP. 1980-09-09 US disclosed