SCHEMBL1047458

SCHEMBL1047458

COc1cc(CCN)c(OC)cc1F

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.69
HTR2A P28223 12/20 0.65
HTR2C P28335 8/20 0.65
HTR2B P41595 6/20 0.58
HTR1A P08908 1/20 0.57
ADRA2A P08913 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
HTR1B P28222 1/20 0.57
HTR7 P34969 1/20 0.57
HTR6 P50406 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29473870 1.00 TAAR1 (0.69) TAAR1HTR2AHTR2CHTR2BHTR1A
Hydrochloric Acid SCHEMBL26096716 0.98 TAAR1 (0.67) TAAR1HTR2AHTR2CHTR2BHTR1A
SCHEMBL20562467 0.90 TAAR1 (0.66) TAAR1HTR2AHTR2CHTR2BHTR1A
SCHEMBL34463042 0.90 TAAR1 (0.66) TAAR1HTR2AHTR2CHTR2BHTR1A
SCHEMBL21240834 0.89 TAAR1 (0.83) TAAR1HTR2AHTR2CHTR2B
SCHEMBL20969693 0.88 TAAR1 (0.53) TAAR1HTR2AHTR2CHTR2B
SCHEMBL24163642 0.86 TAAR1 (0.72) TAAR1HTR2AHTR2CHTR2BHTR1A
SCHEMBL30183033 0.86 TAAR1 (0.72) TAAR1HTR2AHTR2CHTR2BHTR1A
SCHEMBL1253319 0.85 TAAR1 (0.77) TAAR1HTR2AHTR2C
SCHEMBL29364056 0.85 TAAR1 (0.77) TAAR1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 305 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
EP-4547250-A1 METHODS AND COMPOSITIONS RELATING TO CONTROLLING PSYCHEDELIC EFFECTS WITH SEROTONIN RECEPTOR MODULATORS Terran Biosciences Inc. (US) 2025-05-07 EP claimed
US-20240335418-A1 SAFER PSYCHOACTIVE COMPOSITIONS ARCADIA MEDICINE, INC. 2024-10-10 US claimed
US-20240197681-A1 METHODS AND COMPOSITIONS RELATING TO PSYCHEDELICS AND SEROTONIN RECEPTOR MODULATORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-06-20 US claimed
WO-2024107445-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES, INC. (US) 2024-05-23 WO claimed
EP-4313030-A1 METHODS AND COMPOSITIONS RELATING TO PSYCHEDELICS AND SEROTONIN RECEPTOR MODULATORS Terran Biosciences, Inc. (US) 2024-02-07 EP claimed
WO-2024006984-A1 METHODS AND COMPOSITIONS RELATING TO CONTROLLING PSYCHEDELIC EFFECTS WITH SEROTONIN RECEPTOR MODULATORS TERRAN BIOSCIENCES INC. (US) 2024-01-04 WO claimed
EP-4264799-A1 CONNECTION UNIT FOR A STATOR, STATOR FOR AN ELECTRIC MACHINE, STATOR ARRANGEMENT, METHOD FOR PRODUCING A STATOR ARRANGEMENT, AND ELECTRIC MACHINE FOR DRIVING A VEHICLE Valeo eAutomotive Germany GmbH (DE) 2023-10-25 EP claimed
EP-4264801-A1 CONNECTION UNIT FOR A STATOR, STATOR ASSEMBLY FOR AN ELECTRIC MACHINE, METHOD FOR PRODUCING A STATOR ASSEMBLY, AND ELECTRIC MACHINE FOR DRIVING A VEHICLE Valeo eAutomotive Germany GmbH (DE) 2023-10-25 EP claimed
WO-2022128424-A1 CONNECTION UNIT FOR A STATOR, STATOR ASSEMBLY FOR AN ELECTRIC MACHINE, METHOD FOR PRODUCING A STATOR ASSEMBLY, AND ELECTRIC MACHINE FOR DRIVING A VEHICLE VALEO SIEMENS EAUTOMOTIVE GERMANY GMBH (DE) 2022-06-23 WO claimed
WO-2022128426-A1 CONNECTION UNIT FOR A STATOR, STATOR FOR AN ELECTRIC MACHINE, STATOR ARRANGEMENT, METHOD FOR PRODUCING A STATOR ARRANGEMENT, AND ELECTRIC MACHINE FOR DRIVING A VEHICLE VALEO SIEMENS EAUTOMOTIVE GERMANY GMBH (DE) 2022-06-23 WO claimed
EP-2884962-B1 PREPARATION OF DESICCATED LIPOSOMES FOR USE IN COMPRESSIBLE DELIVERY SYSTEMS SMARTEK INT LLC (US) 2019-05-01 EP claimed
US-9435816-B2 Deuterium free, stable isotope labeled 2-phenylethylamine hallucinogens and/or stimulants, methods of their preparation and their use CHIRON AS (NO) 2016-09-06 US claimed
US-20150216799-A1 PREPARATION OF DESICCATED LIPOSOMES FOR USE IN COMPRESSIBLE DELIVERY SYSTEMS SMARTEK INTERNATIONAL LLC 2015-08-06 US claimed
EP-2884962-A2 PREPARATION OF DESICCATED LIPOSOMES FOR USE IN COMPRESSIBLE DELIVERY SYSTEMS Smartek International LLC (US) 2015-06-24 EP claimed
US-20140227792-A1 DEUTERIUM FREE, STABLE ISOTOPE LABELED 2-PHENYLETHYLAMINE HALLUCINOGENS AND/OR STIMULANTS, METHODS OF THEIR PREPARATION AND THEIR USE CHIRON A/S (NO) 2014-08-14 US claimed
WO-2014028796-A2 PREPARATION OF DESICCATED LIPOSOMES FOR USE IN COMPRESSIBLE DELIVERY SYSTEMS SMARTEK INTERNATIONAL LLC (US) 2014-02-20 WO claimed
WO-2013014287-A2 DEUTERIUM FREE, STABLE ISOTOPE LABELED 2-PHENYLETHYLAMINE HALLUCINOGENS AND/OR STIMULANTS, METHODS OF THEIR PREPARATION AND THEIR USE CHIRON AS (NO) 2013-01-31 WO claimed
EP-2551675-A1 Deuterium free, stable isotope labeled 2-phenylethylamine hallucinogens and/or stimulants, methods fo their preparation and their use Chiron AS (NO) 2013-01-30 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140227792-A1 DEUTERIUM FREE, STABLE ISOTOPE LABELED 2-PHENYLETHYLAMINE HALLUCINOGENS AND/OR STIMULANTS, METHODS OF THEIR PREPARATION AND THEIR USE PNMT, HTR2C, HTR2A TAAR1 16/4885HTR2A 3/4885HTR2C 2/4885
US-20240197681-A1 METHODS AND COMPOSITIONS RELATING TO PSYCHEDELICS AND SEROTONIN RECEPTOR MODULATORS HTR1A, HTR2A, HTR3A TAAR1 26/4885HTR2A 2/4885HTR2C 5/4885
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A TAAR1 79/4885HTR2A 14/4885HTR2C 42/4885
US-20240335418-A1 SAFER PSYCHOACTIVE COMPOSITIONS HTR6, HTR4, CNR1 TAAR1 22/4885HTR2A 6/4885HTR2C 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.