SCHEMBL10477754

SCHEMBL10477754

CC1C(=O)Nc2cc3[nH]c(-c4ccccc4)nc3cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 4/20 0.46
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 4/20 0.45
HPGD P15428 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
TP53 P04637 3/20 0.45
HSD17B10 Q99714 3/20 0.45
TSHR P16473 2/20 0.45
NFKB1 P19838 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
MAPT P10636 5/20 0.45
GAA P10253 3/20 0.45
GLA P06280 1/20 0.45
HTT P42858 1/20 0.45
GFER P55789 1/20 0.45
RCE1 Q9Y256 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10470299 0.89 PDE3B (0.55) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL10477810 0.85 TCF4 (0.51) NPC1RAB9AKDM4EMAPTCHEK2
SCHEMBL10374413 0.85 PGR (0.47) NPBWR1NPC1RAB9AKDM4EALDH1A1
SCHEMBL10375400 0.84 NPBWR1 (0.43) NPBWR1NPC1RAB9AKDM4EALDH1A1
SCHEMBL10567302 0.83 PDE3B (0.41) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL10567103 0.82 PGR (0.37) MEN1KMT2ASCDPGRPDE4A
SCHEMBL10569181 0.81 NPC1 (0.43) NPC1RAB9APGRPDE4APDE4B
SCHEMBL10567486 0.81 PDE4A (0.35) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL4894393 0.80 FGFR1 (0.53) CHEK2
SCHEMBL10373856 0.79 FBP1 (0.55) TSHRCYP3A4MAPK1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4810801-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them, and use of them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1989-03-07 US disclosed
US-4710510-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them, and use of them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-12-01 US disclosed
EP-0186010-A1 Pyrrolo benzimidazoles, process for their preparation and medicaments containing them Roche Diagnostics GmbH (DE) 1986-07-02 EP disclosed