SCHEMBL10486289

SCHEMBL10486289

CCNC(=O)c1ccc2cc(-c3cccc4c3C3CCC4C3)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.43
TAOK1 Q7L7X3 1/20 0.39
TAOK3 Q9H2K8 1/20 0.39
SLC6A3 Q01959 1/20 0.38
RAB9A P51151 1/20 0.38
CDK8 P49336 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CYP17A1 P05093 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PDK2 Q15119 2/20 0.36
ALOX15 P16050 1/20 0.36
RIPK1 Q13546 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10486277 0.84 MAPK14 (0.45) MAPK14TAOK1TAOK3SLC6A3RAB9A
SCHEMBL10486405 0.84 SLC6A3 (0.50) SLC6A3ALDH1A1CHRNB2CHRNA4
SCHEMBL10486030 0.83 RARG (0.41) SLC6A3KMT2AKDM4EALDH1A1ALOX15
SCHEMBL10486068 0.72 SLC6A3 (0.45) SLC6A3RAB9AALDH1A1CHRNB2CHRNA4
SCHEMBL10486417 0.72 RXRA (0.42) SLC6A3KMT2AKDM4EALDH1A1ALOX15
SCHEMBL14157778 0.71 HPGDS (0.55) RAB9AKMT2ACYP17A1ALDH1A1HDAC3
SCHEMBL3949393 0.69 HDAC3 (0.62) RAB9AKMT2AHDAC3HDAC4HDAC1
SCHEMBL10486412 0.68 RARG (0.44) KMT2AKDM4EALDH1A1ALOX15
SCHEMBL10486065 0.68 SLC6A3 (0.47) SLC6A3ALDH1A1CHRNB2CHRNA4
SCHEMBL13861733 0.67 CHRNB2 (0.41) KDM4EPDK2CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4810694-A SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1989-03-07 US disclosed